Eltoprazine hydrochloride
CAS No. 98206-09-8
Eltoprazine hydrochloride ( DU-28853 hydrochloride )
Catalog No. M16891 CAS No. 98206-09-8
An antiaggressive agent that acts as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
2MG | 29 | In Stock |
|
5MG | 46 | In Stock |
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10MG | 80 | In Stock |
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25MG | 160 | In Stock |
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50MG | 295 | In Stock |
|
100MG | 438 | In Stock |
|
200MG | Get Quote | In Stock |
|
500MG | Get Quote | In Stock |
|
1G | Get Quote | In Stock |
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Biological Information
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Product NameEltoprazine hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionAn antiaggressive agent that acts as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.
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DescriptionAn antiaggressive agent that acts as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.Schizophrenia Phase 2 Clinical
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SynonymsDU-28853 hydrochloride
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PathwayEndocrinology/Hormones
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Target5-HT Receptor
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Recptor5-HT Receptor
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Research AreaNeurological Disease
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IndicationSchizophrenia
Chemical Information
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CAS Number98206-09-8
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Formula Weight256.73
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Molecular FormulaC12H17ClN2O2
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 31 mg/mL; H2O: ≥ 28 mg/mL
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SMILESC1CN(CCN1)C2=C3C(=CC=C2)OCCO3
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Chemical NamePiperazine, 1-(2,3-dihydro-1,4-benzodioxin-5-yl)-, hydrochloride (1:1)
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Sijbesma H, et al. Eur J Pharmacol. 1990 Feb 20;177(1-2):55-66.
2. Jols M, et al. J Pharmacol Exp Ther. 1990 Apr;253(1):284-9.
3. Mos J, et al. Eur J Pharmacol. 1992 Mar 3;212(2-3):295-8.
2. Jols M, et al. J Pharmacol Exp Ther. 1990 Apr;253(1):284-9.
3. Mos J, et al. Eur J Pharmacol. 1992 Mar 3;212(2-3):295-8.
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