Eltoprazine hydrochloride

CAS No. 98206-09-8

Eltoprazine hydrochloride ( DU-28853 hydrochloride )

Catalog No. M16891 CAS No. 98206-09-8

An antiaggressive agent that acts as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 29 In Stock
5MG 46 In Stock
10MG 80 In Stock
25MG 160 In Stock
50MG 295 In Stock
100MG 438 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Eltoprazine hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    An antiaggressive agent that acts as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.
  • Description
    An antiaggressive agent that acts as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.Schizophrenia Phase 2 Clinical
  • Synonyms
    DU-28853 hydrochloride
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    5-HT Receptor
  • Research Area
    Neurological Disease
  • Indication
    Schizophrenia

Chemical Information

  • CAS Number
    98206-09-8
  • Formula Weight
    256.73
  • Molecular Formula
    C12H17ClN2O2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: ≥ 31 mg/mL; H2O: ≥ 28 mg/mL
  • SMILES
    C1CN(CCN1)C2=C3C(=CC=C2)OCCO3
  • Chemical Name
    Piperazine, 1-(2,3-dihydro-1,4-benzodioxin-5-yl)-, hydrochloride (1:1)

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Sijbesma H, et al. Eur J Pharmacol. 1990 Feb 20;177(1-2):55-66.
2. Jols M, et al. J Pharmacol Exp Ther. 1990 Apr;253(1):284-9.
3. Mos J, et al. Eur J Pharmacol. 1992 Mar 3;212(2-3):295-8.
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